Scientific publications 2009

Aurelio L, Valant C, Figler H, Flynn BL, Linden J, Sexton PM, Christopoulos A, Scammells PJ (2009) 3- and 6-Substituted 2-amino-4,5,6,7-tetrahydrothieno[2,3-c]pyridines as A1 adenosine receptor allosteric modulators and antagonists. Bioorg. Med. Chem. 17, 7353-7361. Link to article.

Garcia Lopez MA, Aguado Martinez A, Lamaze C, Martinez-A, C, Fischer T (2009) Inhibition of dynamin prevents CCL2-mediated endocytosis of CCR2 and activation of ERK 1/2. Cell. Signal. 21, 1748-1757. Link to article.

Stewart GD, Valant C, Dowell SJ, Mijaljica D, Devenish RJ, Scammells PJ, Sexton PM, Christopoulos A (2009) Determination of adenosine A1 receptor agonist and antagonist pharmacology using Saccharomyces cerevisiae: Implications for ligand screening and functional selectivity. J. Pharmacol. Exp. Ther. 331, 277-286. Link to article.

Ouertatani-Sakouhi H, El-Turk F, Fauvet B, Roger T, Leroy D, Karpinar DP, Leng L, Bucala R, Zweckstetter M, Calandra T, Lashuel HA (2009) A new class of isothiocyanate-based irreversible inhibitors of macrophage migration inhibitory factor. Biochem. 48, 9858-9870. Link to article.

Micanovic R, Raches DW, Dunbar JD, Driver DA, Bina HA, Dickinson CD, Kharitonenkov A (2009) Different roles of N- and C-termini in the functional activity of FGF21. J. Cell. Physiol. 219, 227-234. Link to article.

Smith NJ, Stoddart LA, Devine NM, Jenkins L, Milligan G (2009) The action and mode of binding of thiazolidinedione ligands at free fatty acid receptor 1. J. Biol. Chem. 284, 17527-17539. Link to article.

Hay DL (2009) Measurement of phosphorylated Extracellular Signal–Regulated Kinase 1 and 2 in an undergraduate teaching laboratory with ALPHAscreen technology. Sci. Signal. 2, tr1. Link to article.

Last updated: September 2011